20 results found for: “muscarinic_receptors”.

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Muscarinic acetylcholine receptor

Muscarinic acetylcholine receptors, or mAChRs, are acetylcholine receptors that form G protein-coupled receptor complexes in the cell membranes of certain...

Last Update: 2020-12-30T17:46:49Z Word Count : 2589 Synonim Muscarinic acetylcholine receptor

Muscarinic antagonist

A muscarinic receptor antagonist (MRA) is a type of anticholinergic agent that blocks the activity of the muscarinic acetylcholine receptor. The muscarinic...

Last Update: 2021-01-12T18:51:59Z Word Count : 1921 Synonim Muscarinic antagonist

Muscarinic agonist

A muscarinic agonist is an agent that activates the activity of the muscarinic acetylcholine receptor. The muscarinic receptor has different subtypes,...

Last Update: 2020-12-02T21:12:43Z Word Count : 611 Synonim Muscarinic agonist

Muscarinic acetylcholine receptor M3

muscarinic acetylcholine receptor, also known as cholinergic/acetylcholine receptor M3, or the muscarinic 3, is a muscarinic acetylcholine receptor encoded...

Last Update: 2021-01-14T09:00:19Z Word Count : 1630 Synonim Muscarinic acetylcholine receptor M3

Muscarinic acetylcholine receptor M2

The muscarinic acetylcholine receptor M2, also known as the cholinergic receptor, muscarinic 2, is a muscarinic acetylcholine receptor that in humans is...

Last Update: 2020-11-26T17:22:54Z Word Count : 2032 Synonim Muscarinic acetylcholine receptor M2

Parasympathetic nervous system

main types of muscarinic receptors: The M1 muscarinic receptors (CHRM1) are located in the neural system. The M2 muscarinic receptors (CHRM2) are located...

Last Update: 2021-01-23T05:43:18Z Word Count : 3757 Synonim Parasympathetic nervous system

Muscarinic acetylcholine receptor M1

The muscarinic acetylcholine receptor M1, also known as the cholinergic receptor, muscarinic 1, is a muscarinic receptor that in humans is encoded by the...

Last Update: 2020-10-19T22:08:47Z Word Count : 1914 Synonim Muscarinic acetylcholine receptor M1

Acetylcholine

five subtypes of muscarinic receptors have been identified, labeled M1 through M5. All of them function as G protein-coupled receptors, meaning that they...

Last Update: 2021-01-20T08:59:07Z Word Count : 4035 Synonim Acetylcholine

Acetylcholine receptor

"cholinergic" receptors. Molecular biology has shown that the nicotinic and muscarinic receptors belong to distinct protein superfamilies. Nicotinic receptors are...

Last Update: 2020-12-27T21:41:53Z Word Count : 1105 Synonim Acetylcholine receptor

Parasympathomimetic drug

or muscarinic receptors. Choline esters Acetylcholine (all acetylcholine receptors) Bethanechol (M3 receptors) Carbachol (all muscarinic receptors and...

Last Update: 2021-01-06T21:11:40Z Word Count : 555 Synonim Parasympathomimetic drug

Muscarinic acetylcholine receptor M4

cerebral cortex. Muscarinic acetylcholine receptors possess a regulatory effect on dopaminergic neurotransmission. Activation of M4 receptors in the striatum...

Last Update: 2020-12-01T20:05:18Z Word Count : 1842 Synonim Muscarinic acetylcholine receptor M4

Muscarine

the blood-brain barrier. Muscarinic agonists activate muscarinic receptors while nicotinic agonists activate nicotine receptors. Both are direct-acting...

Last Update: 2020-12-02T18:49:52Z Word Count : 1872 Synonim Muscarine

Muscarinic acetylcholine receptor M5

The human muscarinic acetylcholine receptor M5, encoded by the CHRM5 gene, is a member of the G protein-coupled receptor superfamily of integral membrane...

Last Update: 2020-12-02T20:12:42Z Word Count : 1466 Synonim Muscarinic acetylcholine receptor M5

Autonomic drug

two types of receptors are involved in neurotransmission, namely nicotinic receptors and muscarinic receptors. These two groups of receptors can bind to...

Last Update: 2019-12-17T19:58:34Z Word Count : 1953 Synonim Autonomic drug

Atropine

contractility. Muscarinic receptor antagonists bind to muscarinic receptors thereby preventing ACh from binding to and activating the receptor. By blocking...

Last Update: 2021-02-13T16:05:51Z Word Count : 3276 Synonim Atropine

Cholinesterase inhibitor

butyrylcholine in the synaptic cleft that can bind to muscarinic receptors, nicotinic receptors and others. This group of inhibitors is divided into two...

Last Update: 2021-01-15T08:57:30Z Word Count : 1008 Synonim Cholinesterase inhibitor

Reflex bradycardia

binds to M2 muscarinic receptors, causing the decrease in heart rate that is referred to as reflex bradycardia. The M2 muscarinic receptors decrease the...

Last Update: 2020-12-17T13:36:21Z Word Count : 387 Synonim Reflex bradycardia

Nicotinic acetylcholine receptor

stimulate the muscarinic acetylcholine receptors but selectively binds to the nicotinic receptors instead. The muscarinic acetylcholine receptor likewise gets...

Last Update: 2021-01-12T19:45:26Z Word Count : 4547 Synonim Nicotinic acetylcholine receptor

Receptor activated solely by a synthetic ligand

and low constitutive activity and this DREADD receptor was named hM3Dq. M1 and M5 muscarinic receptors have been mutated to create DREADDs hM1Dq and hM5Dq...

Last Update: 2021-01-17T04:58:56Z Word Count : 1754 Synonim Receptor activated solely by a synthetic ligand

Bethanechol

choline carbamate that selectively stimulates muscarinic receptors without any effect on nicotinic receptors. Unlike acetylcholine, bethanechol is not hydrolyzed...

Last Update: 2021-02-18T03:31:11Z Word Count : 360 Synonim Bethanechol

Main result

Muscarinic acetylcholine receptor

Muscarinic acetylcholine receptors, or mAChRs, are acetylcholine receptors that form G protein-coupled receptor complexes in the cell membranes of certain neurons and other cells. They play several roles, including acting as the main end-receptor stimulated by acetylcholine released from postganglionic fibers in the parasympathetic nervous system. Muscarinic receptors are so named because they are more sensitive to muscarine than to nicotine. Their counterparts are nicotinic acetylcholine receptors (nAChRs), receptor ion channels that are also important in the autonomic nervous system. Many drugs and other substances (for example pilocarpine and scopolamine) manipulate these two distinct receptors by acting as selective agonists or antagonists.


muscarinic_receptors
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